Compound

OTB-658

Institute of Materia Medica, CAMS & PUMC
Names
Chemical Class:
Oxazolidinone
Drug Target:
Description

Publications. February 2023. Liu H, Zhu H, Fu L, Zhang W, Chen X, Wang B, Guo S, Ding Y, Wang N, Li D, Lu Y. Efficacy of Replacing Linezolid with OTB-658 in Anti-Tuberculosis Regimens in Murine Models.  Antimicrob Agents Chemother. 2023 Feb 16;67(2):e0139922. doi: 10.1128/aac.01399-22. Epub 2023 Jan 9. PMID: 36622240; PMCID: PMC9933650.

 

Publication. August 2021. Guo S, Wang B, Fu L, Chen X, Zhang W, Huang H, Lu Y. In vitro and in vivo activity of oxazolidinone candidate OTB-658 against Mycobacterium tuberculosis  Antimicrob Agents Chemother Aug 16;AAC0097421. doi: 10.1128/AAC.00974-21. Online ahead of print.

Jiang J, Liu Y, Liu X, Zhang D, Huang H, Wang B, Sheng L, Li Y. Simultaneous determination of a novel oxazolidinone anti-tuberculosis OTB-658 and its metabolites in monkey blood by LC-MS/MS. J Chromatogr B Analyt Technol Biomed Life Sci. 2021 Mar 15;1167:122552. doi: 10.1016/j.jchromb.2021.122552. Epub 2021 Jan 18. PMID: 33588346.

OTB-658(N-(((3S,3aS)-8-Fluoro-1-oxo-7-thiomorpholino-3a,4-dihy-dro-1H,3H-benzo[b]oxazolo[3,4-d][1,4]oxazin-3-yl) methyl) acet-amide)

https://pubmed.ncbi.nlm.nih.gov/33588346/

Developer Associations
Institute of Materia Medica, CAMS & PUMC